Lead Discovery Services by BellBrook Labs

Manufacturer BellBrook Labs  |  Available Worldwide
BellBrook Labs Lead Discovery Services

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Lead Discovery Services
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We will work closely with you to define the specific parameters that are important for your lead discovery program and implement the most efficient and cost effective assays and/or kinetic analyses.

Lead Discovery Services Include:

  • Inhibitor Screening – to identify or confirm activity with target
  • Inhibitor Potency Profiling – dose response with target and/or related proteins
  • Residence Time Measurements – determination of koff using ‘jump dilution’ enzymatic assay method
  • Mechanism of Action Studies – kinetic analysis to define mode of inhibition
  • Inhibitor Selectivity Profiling

Example Targets:

  • Protein Kinases
  • Lipid Kinases
  • Carbohydrate Kinases
  • ATPases
  • Methyltransferases
  • Acetyltransferases
  • HDACs
  • GTPases, GAPs, GEFs
  • Phosphodiesterases
  • Helicases
  • Ligases/Synthetases
  • Glycosyltransferases